Cov lus qhia rau kev siv Zolpidem. Kev tshuaj xyuas thiab analogues

Cov txheej txheem:

Cov lus qhia rau kev siv Zolpidem. Kev tshuaj xyuas thiab analogues
Cov lus qhia rau kev siv Zolpidem. Kev tshuaj xyuas thiab analogues

Video: Cov lus qhia rau kev siv Zolpidem. Kev tshuaj xyuas thiab analogues

Video: Cov lus qhia rau kev siv Zolpidem. Kev tshuaj xyuas thiab analogues
Video: Tshuaj zoo rau cov poj niam nyob nruab hlis noj khoom piv 2024, Lub Xya hli ntuj
Anonim

Zolpidem yog dab tsi? Cov lus qhia rau kev siv, cov ntsiab lus thiab cov lus qhia ntawm cov tshuaj no yuav raug tham ntxiv.

Cov lus qhia rau kev siv zolpidem
Cov lus qhia rau kev siv zolpidem

Shape and composition

Zolpidem muaj dab tsi? Cov lus qhia hais tias cov tshuaj nyob rau hauv nqe lus nug muaj xws li ib tug active tshuaj xws li zolpidem hemitartrate (10 mg), nrog rau cov khoom pab. Nws tuaj nyob rau hauv daim ntawv ntawm cov ntsiav tshuaj dawb, uas tau muab tso rau hauv hlwv ntawm 15 daim.

tshuaj kho mob

Cov tshuaj hauv nqe lus nug ua haujlwm li cas? Cov neeg siv phau ntawv qhia li cas txog qhov no? "Zolpidem" nyob rau hauv nws txoj cai ntawm kev ua yog heev ze rau benzodiazepines. Cov tshuaj no muaj peev xwm nthuav tawm hypnotic, anticonvulsant, amnestic, anxiolytic thiab sedative zog.

Cov tshuaj nquag ntawm cov tshuaj muaj kev cuam tshuam ncaj qha rau benzodiazepine receptors ntawm hom thib ob thiab thawj. Nws txhawb kev qhib cov anion neuronal channel nrog kev pab los ntawm GABA receptors, uas tom qab ntawd ua rau muaj kev nce ntxiv ntawm cov tshuaj chlorine.

Cov tshuaj no cuam tshuam kev xaiv. Hauv qhov no, cov nyhuv ntawm kev noj tshuajnyob ntawm qhov koob tshuaj. Yog li, cov tshuaj me me tso cai rau kom ua tiav amnestic, cov leeg nqaij so thiab anxiolytic zog thiab tiv thaiv cov nyhuv hypnotic

Dab tsi yog qhov zoo tshaj ntawm cov tshuaj no? Cov neeg siv phau ntawv qhia li cas txog qhov no? "Zolpidem" accelerates tus txheej txheem ntawm kev tsaug zog thiab txhim kho kev pw tsaug zog zoo. Nws tseem yuav tsum tau muab sau tseg tias tus neeg mob tsis tsaug zog tom qab sawv.

Kinetic Properties

Zolpidem nqus tau li cas? Kev siv cov tshuaj no, lossis nws qhov ntau npaum li cas nyob ntawm qhov qhia. Tom qab li 30-110 feeb, cov tshuaj nquag ntawm cov tshuaj nce mus txog nws qib siab tshaj plaws hauv cov ntshav. Nws yuav luag tag nrho khi rau cov ntshav plasma, thiab nws cov bioavailability yog 70%.

zolpidem cov lus qhia rau kev siv tshuaj xyuas
zolpidem cov lus qhia rau kev siv tshuaj xyuas

Tom qab nkag mus rau hauv daim siab cov ntaub so ntswg, cov tshuaj nkag mus rau cov tshuaj tiv thaiv metabolic, ua rau tsim cov derivatives tsis muaj zog. Qee tus ntawm lawv tawm nrog cov zis thiab kwv yees li 40% nrog cov quav.

Ib nrab-lub neej ntawm cov tshuaj yog 150 feeb. Nrog kev ua txhaum loj hauv daim siab, cov txheej txheem no txuas ntxiv mus txog 10 teev.

Tshuaj "Zolpidem", cov lus qhia rau kev siv, daim duab uas tau nthuav tawm hauv qab no, nkag mus rau hauv niam lub mis.

lawv sau rau dab tsi?

Cov tshuaj hauv nqe lus nug muaj dab tsi? Cov neeg siv phau ntawv qhia li cas txog qhov no? "Zolpidem" yog ib ntsiav tshuaj tsim los normalize pw tsaug zog. Lawv yog siv rau hmo ntuj awakenings, insomnia los yog ntxovnqa.

txwv tsis pub siv

Zoo li txhua yam tshuaj, tshuaj Zolpidem, cov lus qhia uas muaj nyob rau hauv ib lub thawv ntawv, muaj nws tus kheej contraindications rau kev siv. Cov tshuaj tsis raug sau tseg rau:

  • ua xua rau zolpidem lossis lwm yam benzodiazepines;
  • mob hnyav lossis mob ua pa tsis ua haujlwm;
  • pw tsaug zog apnea;
  • xeeb tub;
  • mob siab lossis mob raum;
  • lactation;
  • kev tsis txaus siab;
  • tsis muaj hnub nyoog.
  • zolpidem cov lus qhia rau kev siv yees duab
    zolpidem cov lus qhia rau kev siv yees duab

Nws tseem yuav tsum tau muab sau tseg tias cov neeg uas muaj kev nyuaj siab, nrog rau cov neeg haus cawv, cov neeg quav yeeb quav tshuaj thiab raug kev txom nyem los ntawm lwm hom kev quav tshuaj, yuav tsum ceev faj tshwj xeeb thaum noj cov tshuaj nug. Txwv tsis pub, qhov no yuav ua rau tus neeg mob qhov xwm txheej nyuaj dua.

Cov lus qhia rau kev siv

Zolpidem hauv daim ntawv ntsiav tshuaj tsuas yog yuav tsum tau noj thaum mus pw. Tus qauv npaum li cas ntawm cov tshuaj no yog 10 mg ib hnub twg. Rau cov neeg laus, thawj koob tshuaj yuav yog 5 mg. Yog tias xav tau ceev, nws tuaj yeem ua ob npaug.

Qhov siab tshaj plaws txhua hnub ntawm "Zolpidem" yog 10 mg. Lub sijhawm siv nws yuav tsum tsis txhob ntau tshaj ib hlis.

Rau cov neeg uas muaj kev ntxhov siab tsis zoo, cov kws kho mob pom zoo kom siv cov tshuaj rau 2-5 hnub, thiab rau cov xwm txheej insomnia - 14-21 hnub.

Yog tias kev kho mob nrog Zolpidem txuas ntxiv rau ob peb hnub, tom qab ntawdtshuaj tuaj yeem nres sai. Yog tias kev kho mob ntau tshaj li ib lub lis piam, tom qab ntawd cov koob tshuaj yuav tsum tau txo qis kom tsis txhob muaj qhov tshwm sim tsis xav tau.

Side Effects

Zolpidem ua li cas rau cov neeg mob? Cov lus qhia rau kev siv, kev tshuaj xyuas hais tias feem ntau cov tshuaj hauv nqe lus nug tsis ua rau muaj kev cuam tshuam tsis zoo. Txawm li cas los xij, muaj cov xwm txheej thaum, tawm tsam keeb kwm yav dhau los ntawm kev siv cov tshuaj no, tus neeg mob tseem hnov txog cov teebmeem hauv qab no:

  • xeev siab, tsaug zog, ntuav, mob taub hau, raws plab;
  • paradoxical insomnia, mob plab, arousal;
  • kiv taub hau, npau suav phem, anterograde amnesia (qhov kev pheej hmoo ntawm kev tsim cov tom kawg yog ncaj qha proportional rau cov tshuaj noj).

Nws tseem yuav tsum tau muab sau tseg tias tsis tshua muaj Zolpidem ua rau cov kev tshwm sim hauv qab no:

zolpidem cov lus qhia rau kev siv tshuaj
zolpidem cov lus qhia rau kev siv tshuaj
  • chim siab, tsis meej pem, dysphoria, aggression;
  • kev coj cwj pwm txawv txawv, kev xav tsis zoo, kev quav yeeb tshuaj;
  • pob khaus, mob siab, hyperhidrosis, siab siab enzymes, angioedema;
  • leeg tsis muaj zog, khaus khaus, txo qis kev sib deev, khaus khaus;
  • ataxia, diplopia.

Cov mob ntau dhau

Cov tsos mob dab tsi ntawm kev noj tshuaj ntau dhau tuaj yeem ua rau cov tshuaj "Zolpidem"? Cov lus qhia rau kev siv qhia tias yog cov tshuaj nyob rau hauv nqe lus nug raug tsim txom los yog ua yuam kevnqos tau ntau yam tshuaj, tus neeg mob yuav ntsib: tsis meej pem, ataxia, ua pa nyuaj, txo cov ntshav siab, coma thiab lethargy.

Thaum noj tshuaj ntau dhau, tus neeg mob yuav tsum ntuav kom sai li sai tau (hauv ib teev). Tsis tas li ntawd, tus neeg raug tsim txom yuav tsum tau muab cov enterosorbents.

Thaum tus neeg mob tsis nco qab, ces nws lub plab yuav tsum tau ntxuav nrog kev sojntsuam, thiab kho cov tsos mob kuj tau ua.

Sib tham nrog lwm yam cuab yeej

Puas puas kam noj Zolpidem nrog lwm cov tshuaj? Cov lus qhia rau kev siv (tsuas yog ib tus kws kho mob uas muaj kev paub dhau los yuav tsum sau daim ntawv xaj rau kev yuav cov tshuaj no) hais tias cov tshuaj xws li Ketoconazole tuaj yeem yuav luag ob npaug ntawm ib nrab ntawm lub neej ntawm cov tshuaj. Tsis tas li ntawd, cov tshuaj no tuaj yeem ua rau muaj kev nyuaj siab CNS.

Kev siv tshuaj sib xyaw nrog cawv feem ntau ua rau muaj kev tawm suab ntawm cov tshuaj, nrog rau nws cov tshuaj ntau dhau.

Cov tshuaj "Rifampicin" ua rau kom cov metabolism sai sai, txo cov txiaj ntsig thiab kev xav ntawm cov tshuaj noj.

zolpidem cov lus qhia rau kev siv hauv cov ntsiav tshuaj
zolpidem cov lus qhia rau kev siv hauv cov ntsiav tshuaj

teem caij ceev faj

Cov tshuaj twg yuav tsum tau sau tshuaj Zolpidem nrog ceev faj heev? Cov lus qhia rau kev siv (analogues ntawm cov tshuaj tau teev tseg hauv qab no) qhia tias cov txiaj ntsig ntawm kev kho tuaj yeem ua rau tsis zoo yog tias cov tshuaj hauv nqe lus nug suav nrog:

  • anxiolytics, barbiturates, antiepileptics thiab narcotic analgesics;
  • hypnotics, tshuaj tiv thaiv kev puas siab puas ntsws, centrally acting antitussives thiab antidepressants;
  • tshuaj tiv thaiv kab mob nrog cov nyhuv sedative, tshuaj rau cov tshuaj loog dav dav;
  • Pizotifen, Baclofen thiab Thalidomide.

Nws tseem yuav tsum tau muab sau tseg tias thaum cov tshuaj no ua ke nrog Buprenorphine, kev pheej hmoo ntawm kev ua pa nyuaj siab tau nce ntxiv.

Cov tshuaj "Zolpidem" nrog "Intraconazole" tau tso cai ua ke, tab sis nrog kev ceev faj heev, vim qhov no cov tshuaj pharmacodynamic thiab pharmacokinetic ntawm thawj tus neeg sawv cev tuaj yeem hloov pauv.

Special Information

Koj yuav tsum paub dab tsi txog Zolpidem? Cov lus qhia rau kev siv (hauv cov ntsiav tshuaj, qhov kev kho no yog muag hauv yuav luag txhua lub tsev muag tshuaj) hais tias nrog kev kho mob ntev (kwv yees li 20-30 hnub), tus neeg mob tuaj yeem tsim kev puas siab puas ntsws lossis lub cev nyob ntawm cov tshuaj. Cov tshuaj tiv thaiv zoo li no tshwj xeeb tshaj yog rau cov neeg uas yav dhau los tau pom kev vam khom ntawm cov dej cawv thiab lwm yam tshuaj. Hauv qhov no, cov neeg mob zoo li no yuav tsum tau tswj xyuas tas li, nrog rau kev saib xyuas lawv lub hlwb thiab lub cev ib ntus.

Nws yuav tsum tau sau tseg tshwj xeeb tshaj yog tias qhov kev pheej hmoo ntawm kev quav tshuaj yog nce ntxiv thaum tus neeg sawv cev hauv nqe lus nug tau ua ke nrog lwm cov tshuaj benzodiazepines.

zolpidem cov lus qhia rau kev siv synonyms
zolpidem cov lus qhia rau kev siv synonyms

Thaum noj Zolpidem, tus neeg mob yuav tsum coj mus rau hauv tus account tias hauv 8 teev tom qab noj tshuaj, nws yuav tsumnyob rau hauv pw tsaug zog zoo, txwv tsis pub nws yuav tsim anterograde amnesia.

Yog tias, tom qab ob peb lub lis piam ntawm kev kho mob, insomnia tseem muaj, tus neeg mob yuav tsum tau rov ntsuas dua. Feem ntau yuav, xws li cov tshuaj tiv thaiv paradoxical yog qhov tshwm sim ntawm kev puas hlwb thawj zaug.

Nyob hauv cov txheej txheem ntawm kev kho mob nrog cov lus nug, tus neeg yuav tsum tsis txhob ua cov haujlwm uas yuav tsum tau ua kom muaj zog ntawm kev mloog, nrog rau kev tsav tsheb.

Qee tus neeg (tshwj xeeb tshaj yog cov neeg laus) tuaj yeem tsim kev coj cwj pwm txawv txawv thiab kev puas siab puas ntsws thaum noj Zolpidem. Hauv qhov no, koj yuav tsum tsis txhob noj tshuaj tam sim ntawd.

Thaum muaj kab mob siab, cov tshuaj nquag tuaj yeem nkag mus rau hauv lub cev, thiab tom qab ntawd ua rau muaj qhov tsis zoo.

Cov tshuaj no yuav tsum tau siv nrog ceev faj heev rau cov neeg laus. Qhov no yog vim qhov tseeb tias lawv muaj kev pheej hmoo siab ntawm kev tsim cov tshuaj sedative thiab cov leeg nqaij so, uas tuaj yeem ua rau ntog thiab raug mob.

Hnub Kawg, cov xwm txheej ntawm kev muag khoom, cia

Vim qhov tseeb hais tias cov tshuaj hauv nqe lus nug yog kev quav tshuaj, koj yuav tsum muaj tus kws kho mob daim ntawv yuav khoom. Nws yog ntshaw kom khaws cov tshuaj no rau hauv qhov chaw uas muaj kev tiv thaiv zoo los ntawm cov menyuam yaus, ntawm qhov kub tsis tshaj 25 degrees. Cov tshuaj muaj lub neej txee ntawm peb xyoos.

Similar txhais tau tias thiab cov ntsiab lus

Cov tshuaj feem ntau rau insomnia, uas yogyog cov analogues ntawm Zolpidem, yog cov hauv qab no: Andante, Donormil, Sondox, Barboval, Zopiclone, Sonmil, Imovan.

Raws li cov ntsiab lus, lawv suav nrog: Hypnogen, Ivadal, Zolsana, Oniria, Snovitel, Sanval, Nitrest.

zolpidem cov lus qhia rau kev siv analogues
zolpidem cov lus qhia rau kev siv analogues

Lactation thiab cev xeeb tub

Cov tshuaj hauv nqe lus nug ntawm cov poj niam cev xeeb tub tsis tau kawm. Txawm li cas los xij, cov txiaj ntsig ntawm kev tshawb fawb uas tau ua nyob rau hauv lub chaw kuaj nas hais tias cov tshuaj no muaj cov nyhuv teratogenic. Hauv qhov no, noj Zolpidem thaum cev xeeb tub yog qhov poob siab heev.

Nws tsis tuaj yeem hais tias cov tshuaj tsaug zog me me tuaj yeem nkag mus rau hauv niam cov kua mis. Yog li, lactation yuav tsum tau nres rau lub sijhawm kho.

Kev tshuaj xyuas ntawm cov neeg siv khoom thiab tus nqi ntawm cov tshuaj

Koj tuaj yeem yuav cov tshuaj Zolpidem hauv yuav luag txhua lub tsev muag tshuaj los ntawm kev nthuav qhia tus kws kho mob cov tshuaj rau tus kws muag tshuaj. Tus nqi nruab nrab ntawm cov tshuaj no (10 ntsiav tshuaj) yog hais txog 820-900 rubles. Cov neeg mob hais tias qhov no yog tus nqi siab rau cov tshuaj tsaug zog. Txawm li cas los xij, cov kws tshaj lij tau tshaj tawm tias tus nqi ntawm cov tshuaj no yog qhov ncaj ncees, vim nws pab tau zoo nrog insomnia thiab pw tsaug zog tsis zoo. Cov neeg siv khoom feem ntau pom zoo nrog cov lus kawg. Lawv hais lus zoo txog cov tshuaj, tab sis tsuas yog lawv noj nws nruj raws li kws kho mob sau ntawv lossis cov lus qhia.

Nyob hauv lawv cov lus, cov neeg mob hais tias tuscov tshuaj tso cai rau lawv tsaug zog ib txwm thiab sai, nrog rau kev pw tsaug zog zoo tom qab muaj kev ntxhov siab. Txawm li cas los xij, cov ntsiav tshuaj Zolpidem kuj muaj qhov tsis zoo. Piv txwv li, lawv tuaj yeem ua rau muaj kev phiv tshuaj, uas feem ntau tshwm sim nrog hypersensitivity rau cov tshuaj nquag ntawm cov tshuaj lossis tsis ua raws li txoj cai. Cov teebmeem tsis zoo tshaj plaws yog: mob taub hau, kiv taub hau, xeev siab thiab hnov lus. Hauv qhov no, tus neeg mob tuaj yeem tsim kev quav tshuaj, tshwj xeeb tshaj yog thaum cov tshuaj sib xyaw nrog cov dej cawv.

Pom zoo: