Aromatase inhibitors: tshuaj xyuas, nqi. aromatase inhibitors hauv bodybuilding

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Aromatase inhibitors: tshuaj xyuas, nqi. aromatase inhibitors hauv bodybuilding
Aromatase inhibitors: tshuaj xyuas, nqi. aromatase inhibitors hauv bodybuilding

Video: Aromatase inhibitors: tshuaj xyuas, nqi. aromatase inhibitors hauv bodybuilding

Video: Aromatase inhibitors: tshuaj xyuas, nqi. aromatase inhibitors hauv bodybuilding
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Anonim

Aromatase inhibitors, lossis blockers, yog ib hom tshuaj kho mob uas siv los txo qis cov tshuaj estrogen hauv cov ntshav thiab nce qib ntawm gonadotropic cov tshuaj hormones thiab testosterone. Cov tshuaj no kuj siv los kho thiab tiv thaiv txiv neej gynecomastia.

aromatase inhibitors
aromatase inhibitors

Aromatase inhibitors hauv bodybuilding feem ntau siv thaum lub voj voog ntawm anabolic steroids rau:

  • nce anabolic cov tshuaj hormones hauv cov ntshav;
  • kev tiv thaiv gynecomastia;
  • tiv thaiv kev kub ntxhov;
  • nce kev nyem (vim tshem tawm qhov tsis zoo ntawm cov tshuaj estrogens);
  • txo cov tshuaj estrogen ntawm lub qe qe-pituitary-hypothalamus axis, ua rau kom rov tsim kho sai.

Tsim kom muaj chav kawm, yuav tsum tau coj mus rau hauv tus account qhov tseeb tias aromatizationTsis yog txhua tus anabolic steroids raug cuam tshuam. Kev siv yog tsim nyog thaum siv cov khoom xws li methandrostenolone, methyltestosterone, testosterone thiab nws cov derivatives. Me ntsis aromatized Halotestin, boldenone.

Efficiency

Tus nqi pheej yig tshaj plaws thiab nyiam aromatase inhibitors (yuav luag zoo ib yam ntawm cov txiv hmab txiv ntoo):

khoom

(lub npe thoob ntiaj teb)

Lub npe (muag los ntawm chaw muag tshuaj) Tus nqi kwv yees Ib daim foos siv prophylactic hauv kev tsim lub cev Thaum gynecomastia tshwm
Exemestane Aromasin 1600 rub. 30 tab. 25 mg txhua 2.5 mg (1/2 ntsiav tshuaj) txhua hnub 25mg ib hnub kom txog thaum cov tsos mob zoo. Tom qab ntawd txo qhov koob tshuaj rau prophylactic.
YLetrozole

Letromara (pharmac.)

Letroza

Estrolet

3200 rub.

1000 rub.

30 tab. 2.5mg txhua 0.5mg (1/5 ntsiav tshuaj) txhua hnub 2.5mg ib hnub kom txog thaum cov tsos mob zoo. Tom qab ntawd txo qhov koob tshuaj tiv thaiv.
YAnastrozole

Selana

"Egistrazol"

"Anastrozole Kabi"

1500 rub.

350 RUB

1300 rub.

28 tab. 1 mg ib 0.5 mg (1/2 ntsiav tshuaj) txhua hnub 1mg ib hnub kom txog thaum cov tsos mob zoo. Kev txo qis ntxiv ntawm cov tshuaj rau prophylactic.

Nws yuav tsum tau muab sau tseg tias qhov nruab nrab ntawm cov tshuaj estrogen yog qhov zoo rau cov leeg nqaij, yog li kev tiv thaiv ntau npaum li cas cuam tshuam rau kev saib xyuas ntawm lub cev tsim nyog ntawm cov txiv neej estrogens.

Course use

Feem ntau cov neeg ncaws pob hauv tsev, siv cov tshuaj aromatase inhibitors, siv cov tswv yim hauv qab no: cov tshuaj siv tsuas yog thaum thawj cov tsos mob ntawm gynecomastia tshwm sim (khaus ntawm lub mis, o, liab). Hmoov tsis zoo, txoj hauv kev no tsis tuaj yeem hu ua qhov zoo.

aromatase inhibitors hauv bodybuilding
aromatase inhibitors hauv bodybuilding

Qhov kev txiav txim siab tshaj plaws yog kuaj estradiol tom qab li kaum hnub ntawm kev siv cov tshuaj anabolic steroids nrog lub neej luv luv (Methandrostenolone, Testosterone Propionate) lossis tom qab peb mus rau plaub lub lis piam ntawm kev siv cov esters ntev (Sustanon, Enanthate, "cypionate "). Tom ntej no, qhov nruab nrab ib feem ntawm "Anastrozole" yog tshuaj - 0.5 mg txhua hnub. Tom qab kaum hnub, kev tswj xyuas ntawm estradiol tau ua tiav thiab cov koob tshuaj raug kho raws li qhov tshwm sim.

Ib qho kev xaiv tsis sib haum yog siv qhov qis thiab nruab nrab ntawm Anastrozole, tsom rau kev xav ntawm tus kheej. Yog hais tias kev nyuaj siab tshwm sim tom qab xws li kev kho mob, erectile kawgmuaj nuj nqi, poob hauv libido, uas txhais tau tias koj yuav tsum tau txo qhov koob tshuaj.

Kev Tshawb Fawb

Qhov tshwm sim ntawm kev lag luam muaj nyob rau hauv pej xeem "Letrazole" coj cov khoom no mus rau pem hauv ntej. Muaj ntau qhov kev ntsuam xyuas uas ua pov thawj qhov ua tau zoo ntawm cov tshuaj no hauv cov txiv neej. Kev taw qhia ntawm cov tshuaj tau nrog los ntawm qhov pom tau nce hauv gonadotropin (LH). Kev noj ntau npaum li cas pib los ntawm 0.02 mg (100 npaug qis dua li qhov kho tau): nrog nws, koj tuaj yeem txo qhov concentration ntawm estrogen los ntawm ib feem peb. 50% ntawm "Letrozole" raug tso tawm ntawm lub cev tsis pub dhau 2-4 hnub, uas tso cai rau koj haus nws txhua hnub. Qhov yooj yim qhov tsis zoo yog nws lub peev xwm los txo cov tshuaj estrogen txawm tias me me.

aromatase inhibitor tshuaj
aromatase inhibitor tshuaj

"Anastrozole" yog qhov nrov hauv kev tsim lub cev: nws tau kawm zoo kawg nkaus hauv cov txiv neej raws li kev txo qis estradiol. Empirically, nws tau pom tias koob tshuaj 1-0.5 mg tuaj yeem txo cov qib estradiol los ntawm kwv yees li 50%. Koj tuaj yeem yuav cov khoom no los ntawm cov neeg muag khoom yuav luag kaum npaug pheej yig dua hauv lub tsev muag tshuaj. Pheej yig "Anastrozole Kabi" pom nyob rau hauv megacities.

Nyob hauv nws phau ntawv, Dr. Mauro G. De Pascale tau sau tias: "Nws xav tias estrogens, tsim los ntawm aromatization ntawm testosterone thiab lwm yam anabolic steroids nyob rau hauv lub hypothalamus thiab lub hlwb, txo cov secretion ntawm luteinizing hormone, thiab. Yog li ntawd, kev tsim cov testosterone. " Gilmann thiab Goodmann qhia tias cov lus tawm tswv yim yog qhib los ntawm cov tshuaj estrogen ntau dua li testosterone. Hauv txoj kev no, nws tau piav qhia tias aromatase inhibitors tuaj yeem txo cov nyhuv inhibitoryCov tshuaj anabolic ntawm kev tso tawm cov tshuaj hormones ntawm tus kheej.

Side Effects

Dab tsi yog qhov phom sij ntawm aromatase inhibitors rau txiv neej? Peb paub tias cov tshuaj estrogen hauv me me muaj txiaj ntsig zoo rau txiv neej lub cev. Cov tshuaj estrogen nce ob qho tib si kev ua tau zoo ntawm chav kawm thiab qhov cuam tshuam ntawm androgen receptors. Tsis tas li ntawd, lawv tus kheej muaj kev tiv thaiv thiab anabolic nyhuv.

aromatase inhibitor nqi
aromatase inhibitor nqi

Qhov tseem ceeb ntawm cov leeg estrogen receptors tau piav qhia meej hauv Anna Wiik cov lus tshaj tawm. Qhov tseeb, koob tshuaj loj ntawm cov blockers tuaj yeem txo qis cov tshuaj estrogen yam tsis tsim nyog, ua rau muaj kev phiv xws li:

  • inhibition ntawm cov leeg loj hlob;
  • mob pob qij txha (arthralgia);
  • kev tsis zoo ntawm kev noj qab haus huv thiab poob hauv libido;
  • kev nyuaj siab;
  • lipid ntshav profile teeb meem (cov roj cholesterol siab);
  • txo pob txha muaj zog.

Kev paub meej, cov tshuaj tiv thaiv zoo dua li Tamoxifen.

Natural inhibitors

Cov hauv qab no sawv tawm:

  • caffeine;
  • resveratrol;
  • zinc;
  • nicotine;
  • apigenin;
  • catechins;
  • eriodictyol.

Daim ntawv thov "Anastrozole"

Dab tsi ntxiv yog aromatase inhibitors zoo rau? Cov tshuaj no tau siv dav hauv kev tsim lub cev. Piv txwv li, "Anastrozole" yuav tsum tau khaws cov dej hauv tib neeg lub cev thiab tiv thaiv qhov tshwm sim ntawm gynecomastia (feem ntau ua ke nrog androgens xws li testosterone thiab dianobol, los yog ua ke nrog.finasteride). Tab sis nyob rau hauv cov ntaub ntawv no, tus neeg ncaws pob kuj tau txais ib tug impressive complex ntawm txwv tsis pub siv tshuaj los ntawm "Lus npe ntawm txwv txoj kev thiab tshuaj", uas kuj muaj lawv tus kheej ntau yam ntawm lwm yam teebmeem.

aromatase inhibitors tshuaj nqi
aromatase inhibitors tshuaj nqi

Kev tswj tsis tau siv "Anastrozole" los ntawm cov neeg ncaws pob uas nyiam, tshwj xeeb, kev tsim lub cev, tuaj yeem ua rau mob caj dab, asthenia, lossis txo qis hauv kev sib koom ua ke, mob taub hau, tsaug zog. Tau kawg, qee zaus cov teeb meem thromboembolic thiab mob stroke tuaj yeem txhim kho.

Ntau ntau tau sau txog Anastrozole hauv cov ntawv nyeem rau cov neeg ncaws pob uas yog tshuaj tsis raug mob. Tab sis tej thaj chaw deb thiab tam sim ntawd los ntawm nws qhov kev txais tos tuaj yeem yog qhov tsis muaj kev cia siab thiab kev tu siab tshaj plaws. Tom qab tag nrho, yog tias koj noj ib ntsiav tshuaj (1 mg) ib hnub twg, koj tuaj yeem tau txais cov tshuaj hormonal surge. Los ntawm txoj kev, qhov tshwm sim no tau pom nyob rau hauv ntau dua 80% ntawm cov neeg siv cov khoom no.

Feem ntau, aromatase inhibitors yog cov tshuaj paub zoo. Cov qauv ntawm peb tiam blockers "Anastrozole" thiab, tom qab ntawd, "Vorozol" thiab "Letrozole", tau tsim ua thawj thiab thib ob kab khoom rau kev kho mob ntawm kev mob qog nqaij hlav cancer mis.

Krizin

Rau cov neeg nqa hnyav, lub khw muag tshuaj kuj muaj 5, 7-dihydroxyflavone ("Kryzin"), uas cov neeg ncaws pob siv cov koob tshuaj ntau heev. Nws muaj anti-aromatase zog thiab yog tsim nyob rau hauv ob daim ntawv - MRM-Chrysin, muaj 500 mg ntawm flawless chrysin ib capsule, thiab SciFit-Chrysin ES, muaj ob zaug. Cov khoom xyaw qis dua.

Cov neeg tsim khoom tsis piav qhia txog cov kev mob tshwm sim, tab sis nws yuav tsum nco ntsoov tias txhua yam tshuaj thiab kev npaj nrog cov tshuaj tiv thaiv aromatase tuaj yeem ua rau muaj kev phom sij loj rau tus neeg ncaws pob lub cev. Tsis tas li ntawd, lawv nyob rau ntawm "Cov Ntawv Qhia Txog Kev Txwv thiab Cov Tshuaj."

Reviews

Ntau tus kws tsim lub cev hais tias, raws li kev paub dhau los ntawm kev siv Letrozole (Femara), lawv tau txiav txim siab tias cov khoom no, daws ib qho teeb meem (nce qib estrogen), ua rau muaj ntau yam teeb meem. Tau kawg, aromatase inhibitors rau txiv neej yog qhov tseem ceeb. Tom qab tag nrho, lub cev (xws li txiv neej) siv estrogens los tswj lub cev tsis muaj zog, lub hlwb ua haujlwm, qib roj cholesterol, cov pob qij txha noj qab haus huv, ligaments, thiab lwm yam.

Cov kis las hais tias estrogen ua rau cov leeg nqaij loj hlob hauv lub cev. Noj 2.5 mg ntawm "Letrozole" ib hnub, lawv pib hnov mob hnyav ntawm articular-ligamentous apparatus thiab ua rau cov kab mob sib kis thiab kis kab mob.

aromatase inhibitors hauv khw muag tshuaj
aromatase inhibitors hauv khw muag tshuaj

Ntau tus neeg ncaws pob ntseeg tias "Letrozole" tsuas yog siv tau los ntawm cov kws tsim lub cev hauv kev npaj rau kev sib tw. Ua tsaug rau nws, lawv tshem tawm cov kua dej ntau dhau hauv lub cev (cov kws tshaj lij tsis muaj kev tu siab rau kev noj qab haus huv rau lub hom phiaj ntawm kev yeej). Lawv zoo siab yuav qhov no aromatase inhibitor. Tus nqi haum rau lawv xwb.

Qee tus neeg ncaws pob hais tias Letrozole muaj txiaj ntsig zoo rau lub cev txawm tias qhov ntau npaum li 0.1-0.5 mg. Lawv tshaj tawm tias nws qhov kev cuam tshuam thib ob tsis phem dua li lwm tus.inhibitors thiab tus qauv rau hom tshuaj no. Lawv paub tseeb tias, raws li cov kev xav tau, cov khoom lag luam rov tsim lub ntim ntawm cov noob qes sai dua Tamoxifen thiab Clomid. Lawv kuj hais tias aromatase inhibitors tsim nyog tus nqi.

Qee tus neeg ncaws pob tshaj tawm tias txhua tus blocker tuaj yeem siv tau, tab sis muab cov khoom lag luam siab ntawm Letrozole hauv cov koob me me, nws dhau los ua tus pheej yig tshaj plaws.

YAnastrozole

Hnub no "Anastrozole" yog qhov nrov tshaj plaws blocker. Qhov pheej yig tshaj yog suav tias yog "Selana". Qee qhov aromatase inhibitors tsis tshua tshwm sim hauv khw muag tshuaj, piv txwv li, Anastrozole Kabi.

Ntau tus neeg tsis txuag kev noj qab haus huv thiab xaiv qhov zoo.

aromatase inhibitors rau txiv neej
aromatase inhibitors rau txiv neej

Noj "Anastrozole" raws li lawv tus kheej qib ntawm estradiol. Yog li ntawd, qib ntawm estradiol yog thawj zaug kuaj txhawm rau kho qhov feem raws li kev tshuaj xyuas. Qhov nruab nrab cov koob tshuaj classical yog 0.5 mg ib hnub.

Tom qab kaum hnub, kuv yuav tsum tau sim dua. Yog tias qib ntawm estradiol yog tus qauv, cov koob tshuaj tuaj yeem raug txo mus rau 0.5 mg ob zaug hauv ib lub lis piam. Yog tias nws tseem siab, kev txais tos yuav tsum txuas ntxiv mus. Thiab yog li nws yuav tsum tau ua kom txog thaum qib ntawm estradiol rov qab los.

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