"Baclosan": cov lus qhia rau kev siv, indications, muaj pes tsawg leeg, analogues, phiv

Cov txheej txheem:

"Baclosan": cov lus qhia rau kev siv, indications, muaj pes tsawg leeg, analogues, phiv
"Baclosan": cov lus qhia rau kev siv, indications, muaj pes tsawg leeg, analogues, phiv

Video: "Baclosan": cov lus qhia rau kev siv, indications, muaj pes tsawg leeg, analogues, phiv

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Hauv cov lus qhia rau kev siv, cov ntsiav tshuaj "Baclosan" raug xaiv los ua lub hauv paus ua haujlwm rau cov leeg nqaij. Lawv txo cov excitability ntawm lub davhlau ya nyob twg seem ntawm rhiab afferent fibers thiab suppress intermediate neurons, yog li inhibiting poly- thiab monosynaptic kis ntawm paj hlwb impulses. Tsis tas li ntawd, cov khoom no txo cov kev ntxhov siab ua ntej ntawm cov leeg spindles.

Lub ntsiab lus tseem ceeb ntawm "Baklosan" muaj pes tsawg leeg yog baclofen. Cov tshuaj muaj qhov nqus tau siab. Nws qhov siab tshaj plaws hauv cov ntshav tau mus txog 2-3 teev tom qab noj tshuaj. Cov tshuaj yog sai absorbed los ntawm lub digestive system. Tshem tawm ntawm lub cev los ntawm lub raum. Cov tshuaj txo qis convulsions, txo cov suab nrov ntawm cov leeg pob txha, vim qhov kev xav ntawm cov ceg tawv kuj txo qis.

baklosan thiab cawv
baklosan thiab cawv

Kev piav qhia thiab khaws cia

ntsiav tshuaj "Baklosan" muaj ib puag ncig biconvex zoo li, dawb. Lawv raug tso tawm hauv ob koob tshuaj: 10 mg (muaj kev pheej hmoo sib faib), 25 mg. Lawv tau ntim rau hauv polypropylene hub ntawm 50 daim, uas tau ntim rau hauv ib lub thawv ntawv. Lawv tso tshuaj yam tsis tau kws kho mob sau ntawv.

Lub txee lub neej ntawm cov tshuaj yog 5 xyoos. Nws yuav tsum tau muab cia rau hauv qhov chaw qhuav thiab tsauskub tsis qis dua +25 ° C, deb ntawm cov menyuam yaus.

Kev qhia

Baklosan ntsiav tshuaj muaj cov lus qhia hauv qab no rau kev siv:

  • cerebral palsy;
  • ntau yam sclerosis;
  • mob hlwb raug mob;
  • kab mob ntawm tus txha caj qaum ntawm kev raug mob, degenerative thiab kis kab mob;
  • yuav haus cawv;
  • stroke;
  • mob ntawm lub paj hlwb;
  • meningitis.

Feem ntau, cov kws tshaj lij tau sau tshuaj rau ntau yam kev raug mob, pob txha, dislocations thiab pathologies ntawm tus txha caj qaum. Cawv thiab Baklosan (qhov no tau qhia hauv cov lus qhia rau kev siv) tsis sib xws.

Cov tshuaj yuav tsum tau noj nrog zaub mov. Cov ntsiav tshuaj yog ntxuav nrog dej. Pib kev kho mob nrog 5 mg peb zaug ib hnub twg, koob tshuaj yog nce txhua peb hnub. Tus nqi ntawm cov tshuaj tau nce mus txog thaum tus neeg mob pom tias muaj kev txhim kho tseem ceeb. Cov koob tshuaj tsuas yog nce los ntawm kws kho mob, qee qhov tshwj xeeb nws tuaj yeem ncav cuag 25 mg. Kev tshem tawm ntawm "Baklosan" yuav tsum tau pom zoo nrog tus kws kho mob tuaj koom. Qhov siab tshaj plaws txhua hnub koob tshuaj yog 100 mg.

Side results

tshem tawm ntawm baklosan
tshem tawm ntawm baklosan

Cov kev mob tshwm sim ntawm Baklosan tsis tshua tau sau tseg. Nrog kev saib xyuas zoo, cov tshuaj yuav tsum tau noj los ntawm cov neeg laus uas muaj kev cuam tshuam rau cov khoom ntawm cov tshuaj. Tej yam tshwm sim:

  • xeev siab thiab ntuav;
  • cem quav thiab raws plab;
  • qaug zog thiab kiv taub hau;
  • puffiness;
  • urinary incontinence;
  • kev nyuaj siab;
  • drowsy;
  • xwb;
  • ncauj qhuav.

Cov tshuaj yog tsim nyob rau hauv daim ntawv ntawm me me biconvex ntsiav tshuaj. Lub ntsiab tseem ceeb ntawm cov tshuaj yog, raws li twb tau hais lawm, baclofen. Cov lus qhia rau kev siv rau Baklosan qhia tias cov khoom xyaw ntxiv yog: qos yaj ywm starch, talc, magnesium stearate, gelatin thiab lactose.

Ntau tshaj

Kev siv tshuaj ntau dhau ua rau nws tus kheej nrog cov tsos mob hauv qab no:

  • mob hnyav mob ntshav siab;
  • kev nyuaj siab;
  • tsis meej;
  • coma (nyob rau hauv rooj plaub uas tsis nco qab, cov leeg nqaij hypotension tuaj yeem pom txog 72 teev).

Raws li cov lus qhia rau kev siv Baklosan, yog tias muaj tshuaj lom nrog cov tshuaj thiab cov tsos mob ntawm cov tsos mob saum toj no, cov tshuaj diuretics yuav tsum tau muab rau tus neeg mob tam sim ntawd, pom zoo haus dej kom ntau. Yog tias pom tias ua pa tsis zoo, ces yuav tsum tau muab cov txheej txheem rau lub ntsws ua pa.

Cov lus qhia tshwj xeeb

Yog tias Baclosan tau muab rau tus neeg mob ntshav qab zib mellitus lossis kab mob siab, tom qab ntawd nws yuav tsum tau saib xyuas cov haujlwm tshwj xeeb ntawm cov enzymes - daim siab transaminases, nrog rau cov ntshav qabzib thiab alkaline phosphatase.

Raws li cov lus qhia rau cov tshuaj, rau lub sijhawm ntawm kev kho mob, txhua tus neeg siv yuav tsum tsis txhob ua cov haujlwm txaus ntshai uas yuav tsum muaj lub siab xav thiab lub cev muaj zog, ua kom muaj zog ntxiv.

Qhov tseem ceeb ntawm kev quav tshuaj

Kev kho tsis yog tshuaj nyob rau hauv txoj haujlwm physics. Chemically, tus neeg sawv cev tsis txaus ntshai, txawm li cas los xijBaclofen ua cov tshuaj ua haujlwm tuaj yeem ua rau lub hlwb xav tau rau kev siv cov tshuaj txuas ntxiv.

Nws paub tias Baklosan tuaj yeem ua rau muaj txiaj ntsig zoo los ntawm lwm cov tshuaj, vim li no, cov neeg siv tshuaj yeeb muaj peev xwm siv cov tshuaj no los txhim kho cov nyhuv ntawm cov tshuaj narcotic. Qee zaum, lawv sim ua kom cov leeg nqaij so nrog cawv, uas ua rau tuag taus.

Tolperison

Baklosan cov lus qhia rau kev siv
Baklosan cov lus qhia rau kev siv

Cov khoom tseem ceeb yog tolperisone hydrochloride. Cov khoom siv pabcuam - citric acid, lactose acid (mis qab zib), hyprolose, crospovidone, stearic carbonic acid.

Pharmacological action

"Tolperizon" - ib qho analogue ntawm "Baklosan", belongs rau pawg N-cholinolytics. Ib qho tshuaj kho cov leeg nqaij uas muaj kev xaiv cov nyhuv (kev nyuaj siab) ntawm lub caudal ib feem ntawm lub hlwb tsim reticular, muaj anticholinergic central zog. Nws tsis muaj kev cuam tshuam rau qhov peripheral ntawm tib neeg lub paj hlwb. Cov tshuaj yog tus cwj pwm los ntawm qhov tsis muaj zog vasodilating thiab cov nyhuv antispasmodic.

Cov lus qhia rau kev siv

Cov tshuaj tau sau rau hauv cov xwm txheej hauv qab no:

  • Cov kab mob nrog txhav, leeg nqaij spasm thiab dystonia, obliterating kab mob ntawm cov hlab ntsha (thromboangiitis obliterans thiab atherosclerosis ntawm cov hlab ntsha ntawm sab sauv thiab sab qis, mob ntshav qab zib angiopathy, Raynaud's syndrome).
  • Cerebral and spinal palsy (kev cog lusceg, leeg nqaij spasm thiab hypertonicity, spinal automatism).
  • Lub cev muaj zog uas ua rau muaj kev puas tsuaj rau kev sib txuas ntawm subcortical-thalamic thiab basal ganglia.
  • Tus kab mob me me, kev mob ntawm cov hlab ntshav tom qab thrombotic venous thiab lymphatic ncig, trophic ulcers ntawm sab ceg, qaug dab peg, hypertonicity, ua ke nrog kev ua txhaum ntawm cov leeg nqaij ntawm ntau hom, nrog rau encephalopathy, uas muaj vascular. etiology.
baclosan phiv
baclosan phiv

koob tshuaj, contraindications thiab overdose

Cov tshuaj tau noj hauv qhov ncauj (tsis hais txog kev noj zaub mov) nrog dej. Thawj koob tshuaj rau cov neeg laus yog 50 mg ob lossis peb zaug hauv ib hnub. Maj mam nce nws, nqa mus txog 150 mg. Lub sijhawm ntawm chav kawm yog txiav txim los ntawm tus kws kho mob, nws nyob ntawm qhov xwm txheej ntawm cov kab mob thiab nws qhov hnyav.

Cov tshuaj yuav tsum tsis txhob noj rau hauv cov xwm txheej hauv qab no: myasthenia gravis, hnub nyoog qis dua 1 xyoos, hypersensitivity, thiab thaum cev xeeb tub thiab lactation.

Kev noj ntau dhau ntawm cov khoom tsis yog lom (tolperisone) tuaj yeem ua rau muaj kev ntxhov siab hauv tus neeg mob (tshwj xeeb yog menyuam yaus), ua pa tuag tes tuag taw, convulsions (tonic thiab cyclic), ataxia.

Theizalud

baclosan ntsiav tshuaj
baclosan ntsiav tshuaj

Cov lus qhia rau kev siv "Tizalud" analogue ntawm "Baklosan":

  • mob nqaij leeg vim kev puas tsuaj rau tus txha caj qaum, nrog rau kev phais mob (lub sijhawm tom qab phais);
  • skeletal nqaij spasm hauv cov kab mob neurological: tshaj tawmsclerosis, myelopathy, degenerative kab mob ntawm tus txha caj qaum, mob stroke).

Contraindication: rhiab heev rau cov tshuaj nquag - tizanidine. Nrog ceev faj, cov tshuaj tau raug sau tseg rau kev ua txhaum ntawm kev ua haujlwm ntawm lub raum thiab lub siab. "Tizalud" yuav tsum tsis txhob siv thaum cev xeeb tub, tshwj tsis yog nyob rau hauv cov xwm txheej uas qhov kev kwv yees tau txais txiaj ntsig rau leej niam tshaj qhov kev hem thawj rau tus menyuam hauv plab. Yog tias koj yuav tsum siv cov tshuaj thaum lactation, koj yuav tsum tsis txhob pub mis niam.

Mydocalm

baclosan analogues
baclosan analogues

"Mydocalm" yog cov leeg nqaij so ntawm lub hauv paus ua haujlwm. Cov lus qhia siv rau Baklosan thiab Mydocalm yog qhov zoo sib xws. Cov tom kawg yog muab raws li hauv qab no:

  • muscle hypertonicity;
  • nrog rau cov leeg nqaij dystonia (nrog rau thaum yau) encephalopathy;
  • muscle spasm;
  • CP;
  • neurological organic thiab degenerative kab mob nyob rau hauv uas striated nqaij tone raug soj ntsuam.
baclosan qhia
baclosan qhia

Qhov txiaj ntsig tseem ceeb ntawm Mydocalm yog los so cov leeg nqaij thiab daws cov teeb meem ntawm cov leeg nqaij uas tshwm sim los ntawm ntau yam. Qhov kev ua tau zoo ntawm cov tshuaj tau raug pov thawj hauv kev tshawb nrhiav qhov muag tsis pom. Qhov kev txiav txim ntawm "Mydocalm" yog lub hauv paus, vim tias cov txiaj ntsig tau ua ncaj qha rau ntawm lub hlwb, Cov tshuaj muaj contraindications:

  • tus neeg tsis kam lees;
  • mob vwm;
  • psychosis;
  • Parkinson's disease.

Kev siv tshuaj thaum cev xeeb tub yog tso cai tshwj xeeb, thaum txoj kev kho mob siab dua qhov kev pheej hmoo rau tus menyuam.

"Mydocalm" yog noj ntawm qhov ncauj, ntsiav tshuaj yuav tsum tau nqos nrog dej. Thaum pib ntawm koob tshuaj rau tus neeg laus - 50 mg ob lossis peb zaug hauv ib hnub, tom qab ntawd los ntawm kev nce peb zaug hauv koob. Yog tias muaj kev phiv tshwm sim (cov leeg tsis muaj zog, ntshav siab, mob taub hau), koob tshuaj yuav tsum raug txo.

Lwm yam khoom

Lwm cov khoom siv tau zoo ntawm cov tshuaj: txo qis excitability ntawm tus txha caj qaum, stabilizing lub sheaths ntawm receptive thiab lub cev muaj zog fibers, txo qhov txhav thiab cov leeg nqaij. Tsis zoo li lwm yam tshuaj zoo sib xws, "Mydocalm" tsis qhia cov nyhuv sedative, tsis muaj kev cuam tshuam ntau dhau ntawm cov kab mob hematopoietic.

Lwm yam analogues

Nyob hauv lub tsev muag tshuaj koj tuaj yeem pom ntau cov analogues, xws li:

  • "Katadolon";
  • "Memikar";
  • "Memorel";
  • "Mementine".

Katadolon yuav tsum tau saib xyuas zoo. Cov tshuaj no muaj zog txaus, tab sis nws tsis suav hais tias yog tshuaj narcotic. Nws muaj zog analgesic nyhuv. "Baclofen" kuj tseem pab tshem tawm qhov mob, txo cov leeg nqaij. Nrog kev pab los ntawm Memorel ntsiav tshuaj, koj tuaj yeem kho lub siab ib txwm muaj, txhim kho kev nco. "Memantine"muaj raws li cov hmoov, nws pab kom muaj zog.

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