"Flutamide": cov lus qhia rau kev siv, piav qhia ntawm cov tshuaj, analogues thiab kev phiv

Cov txheej txheem:

"Flutamide": cov lus qhia rau kev siv, piav qhia ntawm cov tshuaj, analogues thiab kev phiv
"Flutamide": cov lus qhia rau kev siv, piav qhia ntawm cov tshuaj, analogues thiab kev phiv

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"Flutamide" yog ib qho ntawm cov tshuaj antiandrogenic thiab siv los tshem tawm cov tsos mob ntawm androgenization. Nws muaj peev xwm txo qis cov txheej txheem metabolic ntawm androgenic cov tshuaj hormones thiab ua kom nws cov txiaj ntsig zoo rau cov kabmob uas xav tau kev kho mob. Lub hom phiaj tseem ceeb ntawm cov tshuaj yog kev tawm tsam ntawm cov txiv neej cov tshuaj hormones, rau kev kho mob ntawm cov kab mob tshwm sim los ntawm nws qhov ntau dhau.

Flutamide cov lus qhia rau kev siv
Flutamide cov lus qhia rau kev siv

tshuaj muaj txiaj ntsig

Cov tshuaj "Flutamide-250" yog siv rau hauv kev kho mob ntawm cov poj niam thiab cov txiv neej nrog cov tsos mob ntawm testosterone ntau lawm, raug kev txom nyem los ntawm qhov tshwm sim tsis zoo thiab tshwm sim ntawm cov tshuaj hormone no. Cov tshuaj uas tsis yog-steroidal inhibit androgen biosynthesis thiab gland secretion, txo qhov tsim ntawm gonadotropin, thiab kuj txo cov concentration ntawm active androgen molecules. Cov tshuaj activates cov txheej txheem metabolic, txhim khu kev ua haujlwm metabolic kom tshem tawm cov tshuaj hormones ntau dhau ntawm lub cev.

Nrog rau pab pawg ntawm cov tshuaj nonsteroidal thiab yog 5-a-reductase antagonist. Kev noj "Flutamide" tsis cuam tshuam rau kev tsim cov gonadotropin hauv cov qog pituitary thiab tsis txo cov kev ua haujlwm gonadotropic.

flutamide nqi
flutamide nqi

Indications rau nkag

Kev ua tau zoo ntawm kev kho mob coj cov nyhuv nyuaj ntawm cov txheej txheem ntawm kev txo qis qib ntawm cov tshuaj hormones nquag. Lub hom phiaj ntawm Flutamid yog dab tsi? Cov lus qhia rau kev siv qhia qhov txo qis, thiab tom qab ntawd inhibition ntawm cov txheej txheem androgenization.

Raws li qhov tshwm sim ntawm kev tsim cov androgens ntau ntxiv, kev ua haujlwm ntawm enzyme 5-α-, uas yog koom nrog hauv kev tsim tawm ntawm daim tawv nqaij thiab pab txhawb kev nkag siab ntawm nws cov receptors rau cov tshuaj hormones, nce. Yog li pib txoj kev loj hlob ntawm idiopathic hirsutism uas xav tau kev kho mob.

Txog thaum tsis ntev los no, nws tau raug sau tseg rau kev kho mob ntawm prostatic hyperplasia hauv cov txiv neej, tab sis tsis ntev dhau los nws cov txiaj ntsig zoo tau tshwm sim, tsom rau kev kho mob ntawm qee yam poj niam kab mob. Nrog hirsutism, alopecia "Flutamide" rau cov poj niam, thaum noj txhua hnub rau peb lub hlis, txo qis qib ntawm cov txiv neej cov tshuaj hormones hauv cov ntshav, thiab cov kab mob no poob lawv qhov hnyav.

Flutamide tshuaj xyuas
Flutamide tshuaj xyuas

Kab mob uas tshuaj qhia

  • Prostate cancer nrog kis ntawm metastases hauv txiv neej.
  • Hirsutism thiab alopecia hauv cov poj niam.
  • Thaum txiv neej raug phais castrated.
  • Hormonal disorders nrog cov tsos mob pob txuv.
  • Yog tias nchuav menyuamcev xeeb tub los yog tsis muaj peev xwm xeeb tub.

Cov lus qhia tseem ceeb yog cov tsos mob qhia tias muaj ntau tshaj ntawm testosterone hauv lub cev. Hauv cov poj niam, qhov no yog cov txiv neej ntau dhau cov plaub hau, taub hau, kev coj khaub ncaws tsis xwm yeem, thiab lwm yam. Tseem muaj cov tshuaj hormone metabolism hauv cov tsos mob zais, xws li anovulation, uterine thiab mammary gland hypoplasia.

Yuav kom kuaj tau qhov tseeb, tus kws kho mob tau sau ib qho kev kuaj ntxiv, uas suav nrog kev tshawb fawb ntxaws txog kev kuaj ntshav rau lub xeev ntawm qib ntawm ntau yam tshuaj hormones hauv lub cev.

flutamide rau cov poj niam
flutamide rau cov poj niam

Kev siv tshuaj ywj pheej, yam tsis muaj kev pom zoo los ntawm tus kws kho mob tuaj koom, tuaj yeem ua rau muaj kev phom sij rau kev noj qab haus huv. Kev kho mob yuav tsum yog kws kho mob nruj me ntsis!

Txoj kev txais tos

Rau cov tshuaj "Flutamide" cov lus qhia rau kev siv qhia txog qhov ua tiav ntawm qhov siab tshaj plaws hauv cov ntshav 2-3 teev tom qab noj, uas qhia txog kev nqus sai ntawm cov tshuaj los ntawm txoj hnyuv. Ib nrab-lub neej yog hais txog 5-6 teev nyob rau hauv cov zis, thiab me ntsis tom qab, tom qab 8-9 teev, cov seem yog tawm. Qhov zoo ntawm kev tso tawm ncaj qha nyob ntawm lub hnub nyoog ntawm tus neeg mob thiab lub xeev ntawm kev noj qab haus huv.

Kab mob nrog cov tsos mob ntawm androgenization hauv cov poj niam xav tau ib tus neeg mus rau kev kho mob. Kev txiav txim siab txog qib, qhov hnyav, qhov chaw ntawm thaj chaw teeb meem thiab lwm yam cuam tshuam rau cov tshuaj noj, feem ntau yog "Flutamide" raug tshuaj thaum noj cov complex. Cov lus qhia rau kev siv qhia tau hais tias noj peb zaug ib hnub twg, ib ntsiav tshuaj, saib sib npauglub sij hawm. Qhov koob tshuaj txhua hnub yog 750 mg, qhov tsawg kawg nkaus ntawm kev kho mob yog rau lub lis piam.

Flutamide 250
Flutamide 250

Kev kho cov tsos mob ntawm androgen yuav tsum tau ua ke nrog qee yam tshuaj tiv thaiv androgenic. Feem ntau, Dexamethasone, Prednisolone thiab lwm yam corticosteroids tau sau tseg hauv txoj haujlwm. Cov txheej txheem sedative kuj tseem siv los txhawb kev ntxhov siab ntawm cov neeg mob uas muaj cov tsos mob pom tseeb tshwm sim los ntawm kev tawm tsam ntawm cov tshuaj hormones.

Txawm tias tsis muaj cov tsos mob cuam tshuam yav dhau los, nws tsis pom zoo kom tshem cov tshuaj ntawm koj tus kheej, rau qhov no koj yuav tsum sab laj nrog tus kws kho mob endocrinologist uas saib xyuas kev txhim kho ntawm tus kab mob. Yuav tsum ua raws li txhua yam tshuaj uas kws kho mob tau sau tseg. Yog tias vim li cas cov ntsiav tshuaj tsis tuaj, ces koj yuav tsum tsis txhob noj ob zaug ntxiv, tab sis tsuas yog txuas ntxiv qhov noj li niaj zaus. Kev hla tshuaj tsis yog phem npaum li kev noj ob zaug ib zaug.

Ib daim foos

Tau hauv daim ntawv tshuaj ntsiav lossis cov ntsiav tshuaj coated. Npaj rau kev tswj qhov ncauj. Cov khoom xyaw nquag yog flutamide 250 mg.

Nyob hauv khw muag tshuaj, "Flutamid" tsuas yog muag los ntawm cov tshuaj.

Khaws rau hauv qhov chaw qhuav thiab txias kom deb ntawm cov menyuam yaus.

Tsim los ntawm Orion Corporation, tuam txhab tshuaj (Finland).

Rau "Flutamid" tus nqi yog los ntawm 1798 txog 1968 rubles ib pob (84 ntsiav tshuaj).

YContraindications

Raws li kev xyaum tau qhia, tsis muaj kev paub txaus hauv kev kho cov poj niam, hauvqhov no feem ntau cuam tshuam txog qhov tsis paub tseeb hauv kev paub txog cov kev mob tshwm sim thiab kev phom sij rau lub siab. Yog li ntawd, txawm tias qhov ua tau zoo, cov tshuaj yuav tsum tau ceev faj, ua raws li cov kws kho mob cov lus pom zoo.

  • Flutamide yuav tsum tsis txhob noj los ntawm cov neeg mob thyroid, siab lossis raum kab mob.
  • Ntau rhiab heev rau cov khoom ntawm cov tshuaj "Flutamide".
  • Contraindications rau mob raum, siab, pancreas.
  • Siv ceev faj rau cov neeg uas nyiam ua rau cov ntshav txhaws thiab muaj kev cuam tshuam ntawm cov hlab plawv.
cov ntsiav tshuaj flutamide
cov ntsiav tshuaj flutamide

Kev sib tham nrog lwm yam tshuaj

Ua ntej siv cov tshuaj, nws raug nquahu kom qhia rau tus kws kho mob tias cov tshuaj twg noj tsis tu ncua. Tus kws kho mob yuav tsum tau coj mus rau hauv tus account qhov kev tsis txaus siab ntawm kev noj cov vitamins, khoom noj khoom haus, mus txog rau kev noj charcoal.

  • "Flutamide", thaum siv ib txhij nrog lwm cov tshuaj, tuaj yeem txhim kho cov nyhuv ntawm cov tshuaj tiv thaiv, yog li nws yog qhov tsim nyog los suav cov tshuaj kom raug, suav nrog kev sib cuam tshuam.
  • Kev haus luam yeeb thiab cawv kuj tuaj yeem hloov pauv cov tshuaj ntawm lub cev. Thaum lub sij hawm nkag mus, nws yuav yog qhov tsim nyog kom tso tseg kev quav yeeb quav tshuaj.
  • Tus kws kho mob yuav tsum tau ceeb toom txog cov kab mob ntshav uas twb muaj lawm.
  • Yog tias koj npaj yuav xeeb tub, nco ntsoov nrog koj tus kws kho mob tham txog kev noj tshuaj ntxiv.
  • Qhia tshuaj tsis haum tshuaj yog paub thiab tam sim no.

Ntau tshaj

Yog tias cov ntsiav tshuaj flutamide tau raug coj mus rau hauv ntau npaum li cas, ces nws yuav tsum tau ntxuav lub plab thiab mus rau tsev kho mob lossis tsheb thauj neeg mob. Qhov tshwm sim ntawm kev noj tshuaj ntau dhau tuaj yeem ua rau muaj qhov tsis txaus ntseeg ntau ntxiv hauv cov tshuaj tiv thaiv kab mob lossis kev tso tseg ntawm gonadotropin ntau lawm, uas yuav ua rau muaj kab mob ntxiv. Yog li ntawd, nws yog ib qho tsim nyog yuav tsum tau ua raws li cov cai thiaj li yuav noj Flutamide, cov lus qhia rau kev siv qhia tias ua raws li kev noj tshuaj thiab kws kho mob cov lus qhia.

Side effect

Tom qab siv tau ntev lawm, cov txiv neej yuav pom cov tsos mob ntawm gynecomastia, mob hauv siab, ua kua dej.

Flutamide contraindications
Flutamide contraindications

Yog cov tsos mob hauv qab no tshwm sim, uas tej zaum yuav yooj yim rau lub cev, kev siv tshuaj yuav tsum tau tham nrog kws kho mob, tshwj xeeb tshaj yog tias qhov no tsis tau tshwm sim ua ntej.

Symptoms of side effects

x

  • Nkauj qab zib.
  • qis libido.
  • Lub mis loj hauv cov txiv neej.
  • xeev kev nyuaj siab.
  • Kev ua txhaum ntawm kev pw tsaug zog thiab tsaug zog.
  • Puffiness.
  • Hloov cov zis xim.
  • Nyob.
  • Cov tshuaj tiv thaiv tsis tshua muaj tshwm sim, tab sis nrog cov tsos mob uas tau teev tseg nws yog qhov zoo dua los qhia rau tus kws kho mob, tej zaum koj yuav tau hloov qee yam hauv txoj hauv kev los kho lossis nres tshuaj.

    Analogues

    Antiandrogens yog ib pab pawg tshuaj uas muaj cov cuab yeej ntawm inhibiting ntau ntau ntawm progesterone,ua rau muaj teeb meem loj rau tus neeg mob. Cov tshuaj uas tsis yog-steroidal hauv qab no tuaj yeem raug ntaus nqi rau "Flutamide" zoo li cov khoom thiab muaj pes tsawg leeg:

    • "Cyproterone" yog cov tshuaj progestogen ntau tshaj plaws nrog kev ua haujlwm antigonadotropic.
    • "Spironolactone" ("Veroshpiron"). Qhov thib ob nrov tshaj plaws tshuaj, hloov los ntawm Flutamide, lub hauv paus ntsiab lus ntawm kev ua yog heev zoo sib xws, es, txawm indistinguishable.

    Ua ntej koj pib noj cov tshuaj ntawm pab pawg no, koj yuav tsum xyuas kom meej tias lub hauv paus ntawm tus kab mob tsis cuam tshuam nrog kev xeeb tub, qog. Kev npaj ua tib zoo xav tau rau txoj hauv kev rau kev kho mob ntawm hyperandrogenism, thiab contraindications thiab tus cwj pwm ntawm txhua tus neeg mob yuav tsum tau coj mus rau hauv tus account. Nws yog ib qho tseem ceeb ntawm tus kws kho mob lub sij hawm los piav qhia meej txog cov tsos mob thiab kev tshwm sim ntawm tus kab mob, npe cov kab mob uas twb muaj lawm, tshwj xeeb tshaj yog tias lawv cuam tshuam nrog lub siab ua haujlwm, tsuas yog nyob rau hauv txoj kev no tus kws kho mob yuav tuaj yeem xaiv kev kho mob sib xyaw ua ke. Nrog Flutamide.

    Flutamide contraindications
    Flutamide contraindications

    Reviews

    Cia peb tham luv luv txog cov lus teb txog qhov ua tau zoo ntawm kev noj tshuaj "Flutamide". Kev tawm tswv yim tuaj yeem tham los ntawm cov neeg uas tau kho. Hauv cov poj niam raug kev txom nyem los ntawm cov tsos mob ntawm hirsutism, normalization ntawm cov plaub hau kev loj hlob tau raug sau tseg. Cov qog sebaceous ntawm daim tawv nqaij uas ua rau pob txuv kuj tau rov ua haujlwm li qub.

    Muaj cov xwm txheej uas Flutamide tsis pab ntau, kev tshuaj xyuas tsis tau lees paub qhov txiaj ntsig tshwj xeeb ntawm kev noj nws, qhov no feem ntau yog vimmisdiagnosis lossis yuam kev hauv daim ntawv thov. Qee cov neeg mob tsis ua tiav kev kho mob ntev ntev vim yog tus nqi ntawm cov tshuaj, nyob rau hauv rooj plaub twg koj tuaj yeem sab laj nrog kws kho mob thiab siv cov tshuaj pheej yig dua kom tsis txhob tso tseg kev kho mob. Tus nqi rau "Flutamide" yog qhov siab heev, thiab qhov no yuav tsum tau coj mus rau hauv tus account, kev kho mob ntev heev thiab yuav xav tau qee qhov pov tseg nyiaj txiag.

    Cov lus qhia tshwj xeeb

    Hauv kev kho mob nyuaj, Flutamide yuav tsum tau noj peb hnub ua ntej pib GnRH agonist kom txo qis qhov tshwm sim ntawm kev phiv. Hauv daim siab tsis ua haujlwm, kev kho mob tsuas yog qhia yog tias qhov no yog tib txoj kev uas daws qhov teeb meem. Kev soj ntsuam ntawm daim siab ua haujlwm yuav tsum tau ua. Muaj me ntsis nce hauv daim siab thaum noj "Flutamide", tab sis tom qab tshem tawm ntawm qhov loj los ua ib txwm muaj. Nrog cov tsos mob tsis xav tau, pom zoo tshem tawm cov tshuaj.

    Kev kuaj kom tsim nyog los ntsuas lub siab ua haujlwm yuav tsum tau ua hauv txhua tus neeg mob ib hlis ib zaug rau thawj 4 lub hlis, thiab tom qab ntawd ua ntu zus lossis thaum thawj cov tsos mob ntawm daim siab ua haujlwm tsis zoo (khaus khaus, tso zis tsaus, tsis qab los noj mov, daj daj., nro nyob rau hauv txoj cai hypochondrium). Rau cov txiv neej kho mob mus sij hawm ntev thaum tsis muaj tshuaj lom neeg los yog kev phais castration, yuav tsum tau kuaj cov phev tsis tu ncua los tswj fertility.

    Kev tshawb fawb tsis tau ua los ntawm kev tsav tsheb thiab cov txheej txheem khiav haujlwm. Tab sis yog tias cov tsos mob no tshwm sim,zoo li kiv taub hau lossis mob taub hau, nws yog qhov zoo dua tsis txhob pheej hmoo thiab tsis tsav.

    Pom zoo: